| Sunday, July 4 |
| 4:30 pm (approx.) |
Bus arrives from Logan Airport, Boston.
Registration (Registration: 2-11 pm Sunday & 8 am-11 pm Monday) |
| 5:30-7:15 pm |
Dinner |
| Evening Session |
Discussion Leader: Thomas R. Beattie |
| 7:20-7:30 pm |
Greeting by Gordon Conference Chairs & Staff |
| 7:30-8:20 pm |
Jon Ellman (UC-Berkeley): From Libraries to Function |
| 8:20-8:35 pm |
Discussion |
| 8:35-9:25 pm |
Jean Gariepy (Univ. of Toronto): SKULL libraries: combinatorial protein libraries with a built-in search engine |
| 9:25-9:40 pm |
Discussion |
| 9:40 pm |
Welcome Reception and Mixer |
| Monday, July 5 |
| 7:30-8:30 am |
Breakfast |
| 8:30 am |
Photograph |
| Morning Session |
Discussion Leader: Timothy F. Herpin |
| 9:20-10:10 am |
Derek Hudson (Biosearch Technologies, Inc.): A Re-Appraisal of Solid-Phase Synthesis Supports |
| 10:10-10:25 am |
Discussion |
| 10:25-11:15 am |
Andy Combs (DuPont Pharmaceutical): Target Directed Libraries, From Lead Identification to Optimization |
| 11:15-11:30 am |
Discussion |
| 11:30-11:45 am |
Break |
| 11:45-12:30 pm |
Arasu Ganesan (National University of Singapore): Combinatorially Driven Natural Product Synthesis |
| 12:30-12:45 pm |
Discussion |
| 12:50-1:50 pm |
Lunch |
| 4:00-6:00 pm |
Poster Session #1 |
| 6:15-7:15 pm |
Dinner |
| Evening Session |
Discussion Leader: Eric M. Gordon |
| 7:30-8:00 pm |
Clemens Richert (Tufts Univ.): Spectrometrically Monitored Selection of Oligonucleotides with Improved Target
Selectivity and Affinity |
| 8:00-8:10 pm |
Discussion |
| 8:10-8:30 pm |
Short Talk (to be chosen from poster presenters)
|
| 8:30-8:40 pm |
Discussion |
| 8:40-9:30 pm |
Sheila DeWitt (Orchid): Chips for Synthesis and Analysis |
| 9:30-9:45 pm |
Discussion |
| Tuesday, July 6 |
| 7:30-8:30 am |
Breakfast |
| Morning Session |
Discussion Leader: John S. Kiely |
| 8:30-9:15 am |
Barry Bunin (AxyS): Efficient Parallel Synthesis |
| 9:15-9:25 am |
Discussion |
| 9:25-9:55 am |
Alan Schwabacher (UW-Milwaukee): Fourier Transform Combinatorial Chemistry |
| 9:55-10:05 am |
Discussion |
| 10:05-10:30 am |
Break |
| 10:30-11:15 am |
Joseph Salvino (RPR): Supported Reagents for Chemical Library Synthesis |
| 11:15-11:25 am |
Discussion |
| 11:25-12:15 pm |
Paul Keifer (Varian Instruments): NMR Analysis Tools for Combinatorial Chemistry |
| 12:15-12:30 pm |
Discussion |
| 12:50-1:50 pm |
Lunch |
| 6:15-7:15 pm |
Dinner |
| Evening Session |
Discussion Leader: Edward W. Petrillo |
| 7:30-8:00 pm |
Yen-Ho Chu (OSU): Electrophoretic Methods for Studying Combinatorial Libraries |
| 8:00-8:10 pm |
Discussion |
| 8:10-8:30 pm |
Short Talk (to be chosen from poster presenters) |
| 8:30-8:40 pm |
Discussion |
| 8:40-9:30 pm |
Steve Kaldor (Eli Lilly): Factors Influencing Combinatorial Chemistry Methods Development in the Pharmaceutical Industry |
| 9:30-9:45 pm |
Discussion |
| Wednesday, July 7 |
| 7:30-8:30 am |
Breakfast |
| Morning Session |
Discussion Leader: Michael A. Poss |
| 8:30-9:15 am |
Michal Lebl (Spyder Instruments): High speed parallel synthesis utilizing tilted centrifugation technique |
| 9:15-9:25 am |
Discussion |
| 9:25-9:55 am |
Karri Michaels (Tufts Univ.): Randomly Ordered Addressable Microarrays |
| 9:55-10:05 am |
Discussion |
| 10:05-10:30 am |
Break |
| 10:30-11:15 am |
Amir Hoveyda (Boston College): High-Throughput Screening and Chiral Catalyst Discovery |
| 11:15-11:25 am |
Discussion |
| 11:25-12:15 pm |
Bing Yan (Novartis): Accelerating the optimization of solid-phase organic reactions for combinatorial chemistry |
| 12:15-12:30 pm |
Discussion |
| 12:50-1:50 pm |
Lunch |
| 4:00-6:00 pm |
Poster Session #2 |
| 6:15-7:15 pm |
Dinner |
| Evening Session |
Discussion Leader: Paul E. Wiedeman |
| 7:30-8:00 pm |
Jack Hodges (Parke-Davis): Second Generation Scavenger Resins |
| 8:00-8:10 pm |
Discussion |
| 8:10-8:30 pm |
Short Talk (to be chosen from poster presenters) |
| 8:30-8:40 pm |
Discussion |
| 8:40-9:20 pm |
Eric Jacobsen (Harvard Univ.): Catalyst Lead Discovery and Lead Optimization by Combinatorial Methods |
| 9:20-9:35 pm |
Discussion |
| Thursday, July 8 |
| 7:00-8:30 pm |
Breakfast |
| Morning Session |
Discussion Leader: Eric Swayze |
| 8:30-9:15 am |
Kevin Burgess (Texas A&M Univ.): Solid Phase Syntheses of Peptidomimetics with Secondary Structures Tailored to Neurtrophin Ligands |
| 9:15-9:25 am |
Discussion |
| 9:25-9:55 am |
Tim Powers (Symyx): Combinatorial Approaches to Homogeneous Catalysis |
| 9:55-10:05 am |
Discussion |
| 10:05-10:30 am |
Election of 2001 Chair and Vice-Chair |
| 10:30-11:15 am |
Sam Gerritz (Glaxo-Wellcome): Strategies for the Solid-Phase Synthesis of Hundreds to Thousands of Discretes |
| 11:15-11:25 am |
Discussion |
| 11:25-12:15 pm |
Shu Kobayashi (Univ. of Tokyo): Organic Synthesis for Library Construction |
| 12:15-12:30 pm |
Discussion |
| 12:50-1:50 pm |
Lunch |
| 4:00-6:00 pm |
Chairman's Reception & Wine Tasting |
| 6:15-7:15 pm |
Banquet |
| Evening Session |
Discussion Leader: Hans Ulrich Stilz |
| 7:30-8:00 pm |
Mike Poss (BMS): Solution- and Solid-Phase Combinatorial Optimization of a Novel Lipid-Lowering Agent |
| 8:00-8:10 pm |
Discussion |
| 8:10-9:00 pm |
Kevin Chapman (Merck): Mixtures: If this is wrong, why does it work so well? |
| 9:00-9:15 pm |
Discussion |
| 9:15 pm |
Closing remarks |
| Friday, July 9 |
| 7:30-8:30 am |
Breakfast |
| 9:00 am |
Bus Departs for Logan Airport, Boston |
