Understanding Key Concepts for Lead Optimization

The Gordon Research Seminar on Medicinal Chemistry is a unique forum for graduate students, post-docs, and other scientists with comparable levels of experience and education to present and exchange new data and cutting edge ideas in modern drug discovery projects.

Topics will include discussion of concepts of lead-likeness and also on the impact of chemical structure on physicochemical properties, pharmacology, pharmacokinetic and toxicology outcomes. The application of cutting edge technologies to drug discovery programs will also be discussed. The focus of this meeting is to explore fundamental principles of contemporary medicinal chemistry coupled with poster presentations representing the various therapeutic areas and target classes of current interest in the biotech and pharmaceutical industries. The principles will be presented in a workshop format, allowing for close interaction between practicing medicinal chemists and participating attendees. Case studies of drug discovery projects will highlight successful approaches taken to deliver clinical candidates. Registration support will be available for participants; please contact the chair for details.