Sunday P.M., August 3, 1997
- 6:00 - Dinner
- 7:15 - Welcome and Introductory Remarks - John Dillon
Session I
Chau-Jun Li, Discussion Leader
- 7:30 - Barry Trost, Stanford University: Molecular Gymnastics of Alkynes Mediated by Ruthenium Catalysts
- 8:15 - Discussion
- 8:30 - Break
- 8:45 - Greg Fu, Massachusetts Institute of Technology: Asymmetric Catalysis with Planar-Chiral Heterocycles
- 9:30 - Discussion
Monday A.M., August 4, 1997
Session 2
Sean Nugent, Discussion Leader
- 8:25 - Announcements
- 8:30 - Paul Grieco, Indiana University: Organic Chemistry in Polar Media
- 9:15 - Discussion
- 9:30 - David Tschaen, Merck & Company, Inc.: Stereoselective Synthesis of alpha-Aryloxy Acids
- 10:05 - Discussion
- 10:15 - Break
Session 3
Terry Rathman, Discussion Leader
- 10:30 - Victor Snieckus, University of Waterloo: From Flatland to Prochiral Metalation. Aiming for New Synthetic Methodologies for Aromatics and Heteroaromatics
- 11:15 - Discussion
- 11:30 - Reinhard Hoffmann, Phillips-Universität Marburg: Ventures into Magnesium Carbenoid (alpha-Haloalkyl-Mg)- Chemistry
- 12:15 - Discussion
- 12:30 P.M. - Lunch
- 4:00 - 6:00 - Poster Session 1
- 6:00 - Dinner
Monday P.M., Session 4
Mike Harmata, Discussion Leader
- 7:15 - Gary Posner, Johns Hopkins University: Asymmetric Diels-Alder Cycloadditions of Electronically Matched 2-Pyrones and Various Dienophiles: Applications in Vitamin D Analog Synthesis
- 8:00 - Discussion
- 8:15 - Break
- 8:30 - Kim Janda, Scripps Research Institute: Recent Developments in Antibody Catalysis
- 9:15 - Discussion
- 9:30 - Marc Snapper, Boston College: Short Talk - New Applications for Olefin Metathesis
- 9:45 - Discussion
- 10:30 - Late Night
Tuesday A.M., August 5, 1997
Session 5
Chris Schmid, Discussion Leader
- 8:15 - Photo Session
- 8:40 - Announcements
- 8:45 - Leo Paquette, Ohio State University: Cascade Reactions in Synthesis; The Squarate Ester-Polyquinane Connection
- 9:30 - Discussion
- 9:45 - John Grosso, Bristol-Myers Squibb Company: Process Development for the Preparation of the Antimigraine Avitriptan
- 10:20 - Discussion
- 10:30 - Break
Session 6
Kay Brummond, Discussion Leader
- 10:45 - Robert Mills, SmithKline-Beecham: A Practical Enantioselective Synthesis of the Potent Endothelin Receptor Antagonists, SB209670 and SB 217242
- 11:20 - Discussion
- 11:30 - Henry Rapoport, University of California-Berkeley: Aza Apical Azabicyclos
- 12:15 - Discussion
- 12:30 P.M. - Lunch
- Tuesday Afternoon -
3rd Annual ORP Golf Classic
1st Annual ORP Tennis Classic
Tuesday P.M., Session 7
John Montgomery, Discussion Leader
- 7:15 - Pierre Sinay, Ecole Normale Supérieure: Selective Reactions in Carbohydrate Chemistry
- 8:00 - Discussion
- 8:15 - Break
- 8:30 - Russell J. Linderman, North Carolina State University: New Chemistry of alpha-Alkoxy Stannanes
- 9:15 - Discussion
- 9:30 - Xumu Zhang, Penn State University: Short Talk - Asymmetric Catalysis Based on New Chiral Monophosphines
- 9:45 - Discussion
- 10:30 - Late Night
Wednesday A.M., August 6, 1997
Session 8
Amy Howell, Discussion Leader
- 8:25 - Announcements
- 8:30 - Alesandro Dondoni, Ferrara University: Stereocontrolled Formylation Reactions and their use in Pseudopeptide and Sugar Synthesis
- 9:15 - Discussion
- 9:30 - Jonathan Walker, Parke-Davis: Development and Demonstration of a Pilot Scale Process for CI-1012 and CI-1013, Members of a New Class of Anti-HIV Compounds
- 10:05 - Discussion
- 10:15 - Break
Session 9
T. V. Rajanbabu, Discussion Leader
- 10:30 - William Crowe, Emory University: Metallacycle-Mediated Carbon-Carbon Bond Forming Reactions
- 11:15 - Discussion
- 11:30 - Bruce Lipshutz, University of California-Santa Barbara: Recent Progress in Organometallic Chemistry
- 12:15 - Discussion
- 12:30 P.M. - Lunch
- 4:00 - 6:00 - Poster Session 2
- 6:00 - Dinner
Wednesday P.M., Session 10
Marc Snapper, Discussion Leader
- 7:15 - Masakatsu Shibasaki, University of Tokyo: Heterobimetallic Asymmetric Catalysts. Developments and Applications
- 8:00 - Discussion
- 8:15 - Break
- 8:30 - David Kingston, Virginia Polytechnic University: Chemical and Biological Studies on Paclitaxel (Taxol®), The Agony and the Ecstasy
- 9:15 - Discussion
- 9:30 - Kay Brummond, West Virginia University: Short Talk - Allenes and Pauson-Khand Cycloadditions
- 9:45 - Discussion
- 10:30 - Late Night
Thursday A.M., August 7, 1997
Session 11
Scott Sieburth, Discussion Leader
- 8:25 - Announcements
- 8:30 - Alexander Klibanov, Massachusetts Institute of Technology: Enzyme Catalysis in Organic Solvents-Rational Control of Enzymatic Stereochemistry by the Solvent
- 9:15 - Discussion
- 9:30 - Donald Hou, Schering-Plough Research Institute: Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D 1 Antagonist Sch 39166
- 10:05 - Discussion
- 10:15 - Break
Session 12
Richard Pariza, Discussion Leader
- 10:30 - Pierre-Jean Colson, Searle Company: Asymmetric Synthesis of ß-Amino Acids
- 11:05 - Discussion
- 11:15 - Harold Moore, University of California-Irvine: Thermal Rearrangements of Cyclobutenones - Synthesis of Highly Condensed Ring Systems
- 12:00 - Discussion
- 12:15 - Katsuhiko Tomooka, Tokyo Institute of Technology: Short Talk - Advances in the [1,2]-Wittig Rearrangement: A Highly Stereoselective C-C Bond Forming Reactions
- 12:30 - Discussion
- 12:40 P.M. - Lunch
- 2:00 - Annual Academic / Industrial Softball Game
- 4:00 - 6:00 - Chair's Reception
- 6:00 - Banquet
Session 13
William Bailey, Discussion Leader
- 7:30 - Chau-Jun Li, Tulane University: Short Talk - Exploring Aqueous Media for Reactions and Synthesis
- 7:45 - Discussion
- 7:50 - Joel Hawkins, Pfizer, Inc.: Asymmetric Aldol Chemistry: New Conditions, Spectroscopic Studies and Pilot Plant Applications
- 8:25 - Discussion
- 8:35 - Break
- 8:50 - John D. Roberts, California Institute of Technology: A Personal Retrospective of Organic Chemistry
- 9:50 - Discussion
- 10:05 - Closing Remarks
Friday, August 8, 1997
- 6:30 A.M. - Breakfast
- 9:00 - GRC Chartered Bus Departs for Boston
|
