SUNDAY |
2:00 pm - 9:00 pm | Arrival and Check-in (Office Closed 6:00 pm - 7:00 pm) |
6:00 pm | Dinner |
7:30 pm - 7:40 pm | Welcome / Introductory Comments by GRC Site Staff and Conference Chair, J. Ramon Vargas (Eastman Kodak Company) |
7:40 pm - 9:30 pm | Synthesis of Heterocyclic Natural Products I |
| Discussion Leader: Richmond Sarpong (University of California, Berkeley) |
7:40 pm - 8:25 pm | Erik Sorensen (Princeton University) "Strategic Applications of Double Cyclizations in Complex Natural Product Synthesis" |
8:25 pm - 8:35 pm | Discussion |
8:35 pm - 9:20 pm | Richard P. Hsung (University of Wisconsin) "Cycloaddition Chemistry of Allenamides" |
9:20 pm - 9:30 pm | Discussion |
MONDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Catalysis in Heterocyclic Chemistry: In Memory of Professor Keith Fagnou (1971-2009) |
| Discussion Leader: Stephen Godleski (College at Brockport, SUNY) |
9:00 am - 9:50 am | John F. Hartwig (University of Illinois) "Catalytic Processes for the Derivatization of Heterocycles" |
9:50 am - 10:00 am | Discussion |
10:00 am | Coffee Break / Group Photo (10:15 am) |
10:30 am - 11:00 am | Sarah E. Reisman (California Institute of Technology) "New Strategies and Methods for the Synthesis of Heterocyclic Natural Products" |
11:00 am - 11:10 am | Discussion |
11:10 am - 11:40 am | Fu-An Kang (Johnson & Johnson PRD) "Palladium Catalyzed Phosphonium Coupling in the Direct C-C Bond Formations of Heterocycles" |
11:40 am - 11:50 am | Discussion |
11:50 am - 12:20 pm | Melanie Sanford (University of Michigan) "Catalytic Reactions for the Synthesis and Functionalization of Heterocycles" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session #1 (Convenor: Richmond Sarpong) |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Synthesis of Biologically Active Heterocycles I |
| Discussion Leader: Mark Behnke (Consultant) |
7:30 pm - 8:00 pm | George S. Sheppard (Abbott Laboratories) "Heterocyclic Dual Inhibitors of the Insulin-Like Growth Factor and Epidermal Growth Factor Receptor Families" |
8:00 pm - 8:10 pm | Discussion |
8:10 pm - 8:30 pm | Short Talk: Dionicio R. Siegel (University of Texas at Austin) "Synthesis of (+)-Complanadine A, an Inducer of Neurotrophic Factor Excretion" |
8:30 pm - 8:35 pm | Discussion |
8:35 pm - 9:20 pm | Matthew Shair (Harvard University) "Towards Syntheses of the Lomaiviticins" |
9:20 pm - 9:30 pm | Discussion |
TUESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | New Methodology for the Synthesis of Heterocyclic Compounds |
| **Location change for this morning's session ONLY:** DiStefano Lecture Hall in the Antone Academic Center |
| Discussion Leader: David Lathbury (AstraZeneca) |
9:00 am - 9:30 am | Annaliese Franz (University of California, Davis) "Enantioselective Synthesis of Substituted Oxindoles and Spirooxindoles" |
9:30 am - 9:35 am | Discussion |
9:35 am - 10:20 am | John A. Murphy (University of Strathclyde) "Highly Reactive Nitrogen Heterocycles - Synthesis and Properties" |
10:20 am - 10:30 am | Discussion |
10:30 am | Coffee Break |
11:00 am - 11:30 am | Jin-Quan Yu (The Scripps Research Institute) "Carbon-Heteroatom Bond Formation from C-H Bonds: en Route to Diverse Heterocycles" |
11:30 am - 11:35 am | Discussion |
11:35 am - 12:20 pm | Kay M. Brummond (University of Pittsburgh) "Exploiting Allenes in the Synthesis of Strained Heterocycles" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 6:00 pm | Free Time |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Dye Chemistry |
| Discussion Leader: Tehshik Yoon (University of Wisconsin-Madison) |
7:30 pm - 8:00 pm | Suning Wang (Queen's University) "Photochromic Organoboron with a Heterocyclic Backbone" |
8:00 pm - 8:10 pm | Discussion |
8:10 pm - 8:30 pm | Short Talk: Shelli R. McAlpine (San Diego State University) "Synthesis of Urukthaplestatin A derivatives" |
8:30 pm - 8:35 pm | Discussion |
8:35 pm - 9:20 pm | Kevin Burgess (Texas A&M University) "Fluorescent Probes for Multiplexed Intracellular Imaging" |
9:20 pm - 9:30 pm | Discussion |
WEDNESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Heterocycles in Molecular Engineering |
| Discussion Leader: Paul L. Ornstein (Eli Lilly) |
9:00 am - 9:30 am | Lelia Cosimbescu (Pacific Northwest National Laboratory) "Tuning Electronic Properties of OLED Materials with the use of Pyridines, Pyrimidines and Triazines" |
9:30 am - 9:35 am | Discussion |
9:35 am - 10:20 am | Pablo Ballester (Institute of Chemical Research of Catalonia (ICIQ) and Catalan Institution for Research and Advanced Studies (ICREA)) "Quantitative Evaluation of Anion-Pi Interactions in Solution" |
10:20 am - 10:30 am | Discussion |
10:30 am - 10:40 am | Business Meeting Part 1: |
| (Nominations for 2011 Vice Chair) |
10:40 am | Coffee Break |
11:10 am - 11:30 am | Short Talk: Matthew J. Cook (Queen’s University Belfast) "Cascade Sigmatropic Rearrangements" |
11:30 am - 11:35 am | Discussion |
11:35 am - 12:20 pm | Jonathan L. Sessler (University of Texas at Austin) "Oligopyrroles: Receptors and Chemosensors for Potentially Hazardous Materials" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session #2 (Convenor: Richmond Sarpong) |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Synthesis of Heterocyclic Natural Products II |
| Discussion Leader: Paul J. Reider (Princeton University) |
7:30 pm - 8:15 pm | Phil S. Baran (The Scripps Research Institute) "Aiming for the Ideal Synthesis" |
8:15 pm - 8:25 pm | Discussion |
8:25 pm - 9:15 pm | Robert K. Boeckman Jr (University of Rochester) "New Methodology for The Asymmetric Synthesis Of Medium Ring Nitrogen Heterocycles Applied To An Approach To Nakadomarin A" |
9:15 pm - 9:25 pm | Discussion |
THURSDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Synthesis of Biologically Active Heterocycles II |
| Discussion Leader: John Macor (Bristol-Myers Squibb R&D) |
9:00 am - 9:30 am | Paul Scola (Bristol-Myers Squibb) "Targeting HCV NS3 Protease" |
9:30 am - 9:40 am | Discussion |
9:40 am - 10:10 am | Catherine Tachdjian (Senomyx, Inc.) "Allosteric Modulators of Human Taste Receptors" |
10:10 am - 10:20 am | Discussion |
10:20 am - 10:50 am | Business Meeting Part 2: |
| (Fill out Conference Evaluation Forms; Discuss future Site & Scheduling preferences; Election of the next Vice Chair) |
10:50 am | Coffee Break |
11:10 am - 11:40 am | Andre Lescarbeau (Infinity Pharmaceuticals) "Synthesis of Heterocyclic A-Ring Analogs of the Veratrum Alkaloid Cyclopamine as Hedgehog Pathway Inhibitors" |
11:40 am - 11:50 am | Discussion |
11:50 am - 12:20 pm | Nicholas Magnus (Eli Lilly and Company) "Pictet-Spengler Based Synthesis of a Bisarylmaleimide" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 6:00 pm | Free Time / Optional Wine Tasting Social (4:00 pm - 6:00 pm) |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Heterocycles in Chemical Ecology |
| Discussion Leader: Thomas W. Bell (University of Nevada, Reno) |
7:30 pm - 8:00 pm | Tappey H. Jones (Virginia Military Institute) "Stereochemistry and Functionality in Ant Venom Alkaloids" |
8:00 pm - 8:10 pm | Discussion |
8:10 pm - 9:05 pm | Jerrold Meinwald (Cornell University) "Heterocyclic Compounds as Messenger Molecules in Biotic Interactions" |
9:05 pm - 9:15 pm | Discussion |
9:15 pm - 9:30 pm | Richmond Sarpong (University of California, Berkeley) Vice Chair’s Closing Remarks |
FRIDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am | Depart |