| SUNDAY |
| 2:00 pm - 9:00 pm | Arrival and check-in |
| 6:00 pm | Dinner |
| EVENING SESSION |
| 7:30 pm | Chair's welcome: Cynthia (Cyd) McClure
Conference business: GRC staff |
| Discussion Leader: Marco Ciufolini (Université Claude Bernard Lyon) |
| 7:45 pm - 8:10 pm | Tim Jamison - Massachusetts Institute of Technology
(Invited short talk)
"Development and Applications of Asymmetric Catalytic Fragment Coupling Reactions" |
| 8:15 pm - 8:40 pm | Marisa Kozlowski - University of Pennsylvania
(Invited short talk)
"Asymmetric Oxidative Biaryl Coupling and Efforts Towards the Calphostins" |
| 8:45 pm | Steven Ley - University of Cambridge
"Development of New Methods for Natural Product Synthesis" |
| 9:30 pm | Chair's Reception (snack bar) |
| MONDAY |
| 7:30 am - 8:30 am | Breakfast |
| 8:25 am - 8:45 am | Photo (the photo will be taken at 8:30) |
| MORNING SESSION |
| Discussion Leader: Julia Kubanek (Emory University) |
| 8:55 am - 9:25 am | Andrea Stierle - Montana Tech of the University of Montana
"Bioactive Metabolites from Acid Mine Waste Extremophiles" |
| 9:30 am - 10:00 am | Haiyin He - Wyeth-Ayerst
"Development of New Antibiotics from AC98 Glycopeptides" |
| 10:05 am - 10:30 am | Coffee |
| MID-MORNING SESSION |
| Discussion Leader: Robin Polt (University of Arizona) |
| 10:30 am - 11:10 am | Frank Davis - Temple University
"Asymmetric Synthesis of Amine Derivatives using Sulfinimines (N-Sulfinyl Imines)" |
| 11:15 am - 11:40 am | Dalibor Sames - Columbia University
"Complex Organic Synthesis via C-H Bond Activation" |
11:45 am - 12:30 pm | Cynthia Burrows - University of Utah
"Chemistry and Biochemistry of Hydantoins formed from DNA Damage" |
| 12:30 pm | Lunch |
| 1:30 pm - 4:30 pm | Free Time |
| 4:30 pm - 6:00 pm | Poster Session 1 |
| 6:00 pm | Dinner |
| | EVENING SESSION |
| Discussion Leader: Harold Mastalerz (Bristol-Myers Squibb) |
| 7:30 pm - 8:05 pm | Fred West - University of Alberta
"Stereoselective Rearrangements of Reactive Intermediates: Versatile Methodology for the Construction of Bioactive Targets" |
| 8:10 pm - 8:45 pm | Margaret Faul - Eli Lilly and Co.
"Chemistry and Biology of Novel Indolocarbazoles" |
| 8:50 pm | Ed Vedejs - University of Michigan
"Synthetic Investigations Directed at Unusual Oxazole-Containing Macrocycles" |
| TUESDAY |
| 7:30 am - 8:30 am | Breakfast |
| MORNING SESSION |
| Discussion Leader: Steve Wittenberger (Abbott Laboratories) |
| 8:45 am - 9:10 am | Dennis Wright - University of Florida (Invited short talk)
"Synthetic Methodologies Based on the Chemistry of Furan" |
| 9:15 am - 9:40 am | Jon Rainier - University of Arizona (Invited short talk)
"Efficient Approaches to Highly Substituted Indoles" |
| 9:45 am - 10:00 am | Rich G. Carter - Oregon State University (Short talk)
"Progress Toward the Total Synthesis of the Spirotoxin Azaspiracid" |
| 10:00 am | Coffee Break |
| MID-MORNING SESSION |
| Discussion Leader: Alison Hulme (University of Edinburgh) |
| 10:25 am - 11:10 am | Margaret Brimble - University of Auckland New Zealand
"Synthetic Studies Towards Natural Products Containing Bis-spiroacetals" |
| 11:15 am - 11:40 am | Steven Diver - SUNY at Buffalo (Invited short talk)
"Progress Toward the Synthesis of Ambewelamide A" |
| 11:45 am - 12:30 pm | Alessandro Dondoni - University of Ferrara
"Synthesis Of Glycoconjugate Bioisosteres" |
| 12:30 pm | Lunch |
| 1:30 pm - 4:30 pm | Free Time |
| 4:30 pm - 6:00 pm | Poster Session 2 |
| 6:00 pm | Dinner |
| | EVENING SESSION |
| Discussion Leader: Lee Latimer (Elan Pharmaceuticals) |
| 7:30 pm - 7:45 pm | Dengming Xiao - Array Biopharma (Short talk)
"Enantioselective Total Synthesis of TMC-69" |
| 7:45 pm - 8:15 pm | Paul Hanson - University of Kansas
"Metathesis Strategies to Diverse Heterocycles" |
| 8:20 pm - 8:45 pm | Brian Stoltz - California Institute of Technology (Invited short talk)
"The Synthesis of Complex Natural Products as a Driving Force for the Discovery and Development of New Reactions" |
| 8:50 pm | Gunda Georg - University of Kansas
"Synthesis and Evaluation of Natural Product-Derived Anticancer Agents" |
| WEDNESDAY |
| 7:30 am - 8:30 am | Breakfast |
| MORNING SESSION |
| Discussion Leader: Leslie Jimenez (Rutgers University) |
| 8:45 am - 9:20 am | Christopher Spilling - University of Missouri, St. Louis
"Asymmetric Synthesis with Chiral Hydroxy Phosphonates" |
| 9:25 am - 9:50 am | Keith Woerpel - University of California, Irvine
"New Synthetic Methods for Stereoselective Synthesis" |
| 9:55 am | Coffee |
| MORNING SESSION |
| Discussion Leader: Debra Bemis (Avon Products, Inc.) |
| 10:20 am - 10:35 am | Horacio Olivo - University of Iowa (Short talk)
"Toward the Synthesis of Aurisides and Callipeltosides" |
| 10:35 am - 11:15 am | Yu-Gui Gu - Abbott Laboratories
"Macrolide Antibiotics, from Erythromycin to Ketolides" |
| 11:20 am - 11:45 am | Mary Cloninger - Montana State University (Invited short talk)
"Heterogeneously Functionalized Dendrimers for the Study of Biological Recognition Events" |
| 11:45 am - 12:30 pm | Laura Kiessling - University of Wisconsin - Madison
"Syntheses and Applications of Natural and Non-natural Glycoconjugates" |
| 12:30 pm | Lunch |
| 1:30 pm - 4:30 pm | Free Time |
| 4:30 pm - 6:00 pm | Poster Session 3 |
| 6:00 pm | Dinner |
| EVENING SESSION |
| Discussion Leader: Karl Hansen (Merck & Co.) |
| 7:30 pm - 7:45 pm | Michael Greco - Johnson & Johnson Pharmaceuticals Research and Development (Short talk)
"Nonpeptide Inhibitors of Cathepsin G. Optimization of a Novel -Ketophosphonic Acid Lead by Structure-Based Drug Design"
|
| 7:45 pm - 8:30 pm | Kathy Parker - SUNY Stony Brook
"Strategies and Methods in Organic Synthesis" |
| 8:40 pm | Paul Reider - Merck & Co.
"Synthesis of NK-1 Receptor Antagonists -- It's Not Nice To Fool Mother Nature!" |
| THURSDAY |
| 7:30 am - 8:30 am | Breakfast |
| MORNING SESSION |
| Discussion Leader: Pat McDougal (Reed College) |
| 8:45 am - 9:20 am | Rebecca Braslau - University of California, Santa Cruz
"Nitroxide Mediated Reactions and Polymerizations" |
| 9:25 am - 10:00 am | Melissa Rewolinski - Pfizer, Inc.
"Novel Methodologies Utilized in the synthesis of Capravirine and Related Compounds" |
| 10:05 am | Coffee Break |
| MID-MORNING SESSION |
| Discussion Leader: Dee Ann Casteel (Bucknell University) |
| 10:30 am - 11:15 am | F. Hal Ebetino - Procter and Gamble
"Bioisosteric Drug Design Based on Natural Product Ligands of G-Protein Coupled Seven Transmembrane Receptors" |
| 11:20 am - 11:35 am | Marvin Hansen - Eli Lilly & Co. (Short talk)
"Practical Synthesis of Trans-2,4-Disubstituted Piperidines" |
| 11:40 am - 12:30 pm | Janine Cossy - Laboratoire de Chimie Organique ESPCI
"Enantioselective Methodologies. Applications to the Synthesis of Heterocyclic Natural Products" |
| 12:30 pm | Lunch |
| 2:00 | Annual Academia-Industry Softball game |
| 6:00 pm | Dinner |
| EVENING SESSION |
| 7:30 pm - 7:45 pm | Conference Business |
| Election of Vice-Chair for 2003
Presentation of Softball Awards |
| Discussion Leader: Rita Majerle (South Dakota State University) |
| 7:50 pm - 8:40 pm | Madeleine Joullié - University of Pennsylvania
"Total Synthesis of Natural Products" |
| 8:50 pm | Eric Jacobsen - Harvard University
"New Asymmetric Catalytic Reactions" |
| FRIDAY |
| 7:30 am - 8:30 am | Breakfast |
| 9:00 am | Departure |
