SUNDAY |
2:00 pm - 9:00 pm | Arrival and check-in |
6:00 pm | Dinner |
7:15 pm | WELCOME And Presentation by Salve Regina Official(s) |
7:30 pm - 9:30 pm | STEREOSELECTIVE SYNTHESIS SESSION 1 |
| Discussion Leader: Ernest Eliel (University of North Carolina) |
7:30 pm - 8:15 pm | Scott Denmark (University of Illinois at Urbana-Champaign)
"New Concepts in Asymmetric Catalysis with Chiral Lewis Bases" |
8:15 pm - 8:30 pm | Discussion |
8:30 pm - 9:15 pm | Thomas Lectka (Johns Hopkins University)
"Asymmetric Catalysis with Zwitterionic Enolates: From b-Lactam Synthesis to Enantioselective Halogenation" |
9:15 pm - 9:30 pm | Discussion |
9:30 pm - 10:30 pm | Reception |
MONDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | NEW ASPECTS OF STEREOCHEMISTRY 1 |
| Discussion Leader: Bruce Maryanoff (Johnson & Johnson) |
9:00 am - 9:40 am | Yoshio Okamoto (Nagoya University)
"Efficient Separation of Enantiomers by HPLC Using Polysaccharide Derivatives as Chiral Stationary Phases" |
9:40 am - 9:50 am | Discussion |
9:50 am - 10:30 am | David Walba (University of Colorado)
"Fluid Conglomerates: Chiral Liquid Crystal Phases from Achiral Molecules" |
10:30 am - 10:40 am | Discussion |
10:40 am | Coffee Break |
11:00 am - 11:20 am | Paul Floreancig (University of Pittsburgh)
"Electrophile Formation under Neutral Conditions: Electron Transfer Initiated Cyclization Reactions" |
11:20 am - 11:30 am | Discussion |
11:30 am - 11:50 am | Matthew Sigman (University of Utah)
"Catalytic Enantioselective Oxidations using Molecular Oxygen" |
11:50 am - 12:00 pm | Discussion |
12:00 pm - 12:20 pm | Andrei Yudin (University of Toronto)
"Development of Selective Nitrogen Transfer Processes" |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session A |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | BIOORGANIC TRANSFORMATIONS |
| Discussion Leader: Melissa Egbertson (Merck) |
7:30 pm - 8:10 pm | Sam Gellman (University of Wisconsin at Madison)
"Structure and Function in Natural and Unnatural Peptides" |
8:10 pm - 8:20 pm | Discussion |
8:20 pm - 8:40 pm | Li Deng (Brandeis University) "Catalytic Asymmetric reactions with modified Cinchona alkaloids" |
8:40 pm - 8:50 pm | Discussion |
8:50 pm - 9:30 pm | Suzanne Walker (Princeton University)
"Chemical Approaches to Study Bacterial Enzymes" |
TUESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | STEREOSELECTIVE SYNTHESIS SESSION 2 |
| Discussion Leader: Chris Senanayake (Sepracor) |
9:00 am - 9:40 am | Erick Carreira (ETH Zürich)
"Studies in asymmetric synthesis" |
9:40 am - 9:50 am | Discussion |
9:50 am - 10:30 am | Dhileep Krishnamurthy (Sepracor)
"Studies Towards the Asymmetric Synthesis of Sibutramine Metabolites" |
10:30 am - 10:40 am | Discussion |
10:40 am | Coffee Break |
11:10 am - 11:50 am | James McNamara (Merck)
"Asymmetric Syntheses of NK-1 Receptor Antagonists" |
11:50 am - 12:00 pm | Discussion |
12:00 pm - 12:20 pm | Robert Gawley (University of Miami) "Recent studies of Chiral Organometallics" |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Optional Workshop on Systematic Definition of Regio- and Stereoselectivity
Scott Denmark (University of Illinois at Urbana-Champaign) |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | CATALYTIC ASYMMETRIC TRANSFORMATIONS |
| Discussion Leader: Carol Ensinger (Biogen) |
7:30 pm - 8:10 pm | Shu Kobayashi (University of Tokyo)
"Efficient Asymmetric Catalysis in Aqueous and Organic Solvents" |
8:10 pm - 8:20 pm | Discussion |
8:20 pm - 8:40 pm | Daesung Lee (University of Wisconsin)
"Construction of Quaternary Carbon Centers by C-H Insertion: Progress toward a Total Synthesis of Guanacastepene A" |
8:40 pm - 8:50 pm | Discussion |
8:50 pm - 9:30 pm | David Evans (Harvard University)
"Asymmetric Synthesis with Chiral Metal Complexes" |
WEDNESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | NEW ASPECTS OF STEREOCHEMISTRY 2 |
| Discussion Leader: Amy Howell (University of Connecticut) |
9:00 am - 9:40 am | Ben Feringa (University of Groningen)
"Control and Amplification of Chirality" |
9:40 am - 9:50 am | Discussion |
9:50 am - 10:30 am | Stefan Matile (University of Geneva)
"Self-Assembly of para-Oligophenyl Rods From Supramolecular Architecture to Function" |
10:30 am - 10:40 am | Discussion |
10:40 am | Coffee Break |
11:10 am - 11:50 am | Kay Brummond (University of Pittsburgh)
"A Catalytic Synthesis of Cross-Conjugated Trienes: A Scaffold for Rapidly Increasing Molecular Complexity" |
11:50 am - 12:00 pm | Discussion |
12:00 pm - 12:20 pm | George O'Doherty (West Virginia University) "Use of the sharpless asymmetric dihydroxylation reaction for the synthesis of 1,2- and 1,3-diols" |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session B |
6:00 pm | Dinner |
7:15 pm - 7:30 pm | Business Meeting |
7:30 pm - 9:30 pm | NATURAL PRODUCT CHEMISTRY |
| Discussion Leader: James Morken (University of North Carolina) |
7:30 pm - 8:10 pm | Francis Fang (Eisai)
"Asymmetric Synthesis of New Anti-Cancer Natural Products" |
8:10 pm - 8:20 pm | Discussion |
8:20 pm - 8:40 pm | Jeff Aubé (University of Kansas) "Asymmetric synthesis of the Dendrobatid alkaloid 251F" |
8:40 pm - 8:50 pm | Discussion |
8:50 pm - 9:30 pm | Dan Yang (University of Hong Kong)
"Catalytic Asymmetric Radical Cyclization Reactions" |
THURSDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | HETEROCYCLIC AND MEDICINAL CHEMISTRY |
| Discussion Leader: Jay McGill (Lilly) |
9:00 am - 9:40 am | André Charette (University of Montreal)
"New methodology for the stereoselective synthesis of substituted piperidines" |
9:40 am - 9:50 am | Discussion |
9:50 am - 10:30 am | Donna Huryn (Wyeth)
"Design and Synthesis of Agents to Treat CNS Disorders" |
10:30 am - 10:40 am | Discussion |
10:40 am | Coffee Break |
11:10 am - 11:50 am | Mikiko Sodeoka (Tohoku University)
"Palladium Aqua or Hydroxo Complex as a Unique Chiral Catalyst" |
11:50 am - 12:00 pm | Discussion |
12:00 pm - 12:20 pm | Sergey Kozmin (University of Chicago)
"New Strategies for Multiparallel and Complex Molecule Synthesis" |
12:30 pm | Lunch |
1:30 pm - 6:00 pm | Free Time |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | CHIROPTICAL METHODS |
| Discussion Leader: Nina Berova (Columbia University) |
7:30 pm - 8:10 pm | Prasad Polavarapu (Vanderbilt University)
"Recently Developed Methods for Determining the Absolute Configuration and Predominant Conformers" |
8:10 pm - 8:20 pm | Discussion |
8:20 pm - 8:40 pm | Richard Taylor (University of Notre Dame) "Conformation-activity relationships in macrolide natural products" |
8:40 pm - 8:50 pm | Discussion |
8:50 pm - 9:30 pm | Koji Nakanishi (Columbia University)
"Stereochemical Aspects of Rhodopsin: CD Studies" |
FRIDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am | Departure |