SUNDAY |
2:00 pm - 9:00 pm | Arrival and check-in |
6:00 pm | Dinner |
7:20 pm | Carol Ensinger (Deciphera Pharmaceuticals, LLC)
Welcome and Introductory Remarks |
7:30 pm - 9:30 pm | NEW REACTIONS AND MACROMOLECULES |
| Discussion Leader: Ann Gelormini (Aventis Pharmaceuticals) |
7:30 pm - 8:30 pm | Pierre Deslongchamps (University of Sherbrooke)
"New General Strategies for the Construction of Complex Steroids and Terpenoids" |
8:30 pm - 9:30 pm | J. Fraser Stoddart (UC-Los Angeles)
"Dynamic Chirality and Topology" |
MONDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | STEREOSELECTIVE SYNTHESIS |
| Discussion Leader: George O'Doherty (West Virginia University)
|
9:00 am - 9:30 am | Hélène Lebel (University of Montreal)
"Activation of Nitrogen Derivatives with Transition Metal Complexes: Towards Stereoselective Processes" |
9:30 am - 10:00 am | Nobuyoshi Yasuda (Merck Research Laboratories) "Preparation of mGluR Agonists" |
10:00 am - 10:30 am | Group Photo and Coffee Break |
10:30 am - 11:15 am | Mark Lautens (University of Toronto)
"Making and Breaking Rings: New Methodology and Applications" |
11:15 am - 12:00 pm | Anthony G.M. Barrett (Imperial College, London)
"Recent Advances in the Total Synthesis of Antibiotics" |
12:00 pm - 12:30 pm | Michael Krische (University of Texas--Austin)
"Enones as Latent Enolates in Catalysis: Discovery of Catalytic C-C Bond Forming Hydrogenations" |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session A |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | "GREEN" CHEMISTRY |
| Discussion Leader: Robert Gawley (University of Arkansas) |
7:30 pm - 8:15 pm | Yian Shi (Colorado State University)
"Organocatalytic Oxidation: Development of Ketone Catalyst for Asymmetric Epoxidation of Olefins with Broad Scope" |
8:15 pm - 9:00 pm | Steve Nolan (University of New Orleans)
"Recent Advances in the Use of N-Heterocyclic Carbene Ligands in Homogeneous Catalysis" |
9:00 pm - 9:30 pm | Ulf Lindström (Lund University, Sweden)
"Towards Synthetic Efficiency in Water - Principles, Strategies and Methods" |
TUESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | BIOORGANIC AND NATURAL PRODUCTS CHEMISTRY |
| Discussion Leader: Fraser Fleming (Duquesne University) |
9:00 am - 9:45 am | John Wood (Yale University)
"Bridged Polycyclic Natural Products: Inspirational Targets for Synthesis" |
9:45 am - 10:15 am | David Varie (Lilly Research Laboratories)
"An Asymmetric Synthesis of a Conformationally Restricted Glutamic Acid Analog" |
10:15 am - 10:30 am | Coffee Break |
10:30 am - 11:15 am | Marvin Miller (University of Notre Dame) |
11:15 am - 12:00 pm | David Williams (Indiana University)
"New Developments for Stereochemical Control in the Synthesis of Marine Natural Products" |
12:00 pm - 12:30 pm | John Roberts (GlaxoSmithKline)
"Novel Syntheses of (3R, 3aS, 6aR)-Hexahydrofuro[2,3-b]furan-3-ol" |
12:30 pm | Lunch |
1:30 pm - 6:00 pm | Free Time |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | NON-SYNTHETIC METHODOLOGY |
| Discussion Leader: Dhileep Krishnamurthy (Boehringer-Ingelheim) |
7:30 pm - 8:15 pm | Peter Wipf (University of Pittsburgh)
"Structural Puzzles in Organic Synthesis" |
8:15 pm - 8:45 pm | Willy Hauck (Groupe NOVAsep)
"Integrating Multicolumn Continuous Chromatography in Global Chiral Syntheses: a Real Alternative" |
8:45 pm - 9:30 pm | Thomas Szyperski (University of Buffalo)
"Rapid Acquisition of Multidimensional NMR Data" |
WEDNESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | STEREOSELECTIVE SYNTHESIS |
9:00 am - 9:45 am | Jeff Johnston (Indiana University)
"The Development of New Reactions and Reagents for Alkaloid Total Synthesis" |
9:45 am - 10:15 am | Bridget Rohde (Abbott Laboratories) "Synthesis of a Novel Farnesyl Transferase Inhibitor, ABT-100; Selective Preparation of a Stereogenic Tertiary Carbinol" |
10:15 am - 10:45 am | Coffee Break |
10:45 am - 11:15 am | Cathy Crudden (Queens' University)
"Catalytic Asymmetric Synthesis Via Main Group Organometallics" |
11:15 am - 12:00 pm | Matt McIntosh (University of Arkansas)
"Claisen and Aldol Approaches to the Eunicellin Diterpenes" |
12:00 pm - 12:30 pm | Dirk Trauner (UC-Berkeley)
"Stereoselectivity in Electrocyclizations" |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session B |
6:00 pm | Dinner |
7:15 pm - 7:30 pm | Business Meeting |
7:30 pm - 9:30 pm | MACROMOLECULAR CHEMISTRY |
| Discussion Leader: Michael Palucki (Merck Research Laboratories) |
7:30 pm - 8:15 pm | Lin Pu (University of Virginia)
"Fluorescent Sensors in Chiral Recognition" |
8:15 pm - 8:45 pm | Tom Rovis (Colorado State University)
"Chiral Nucleophilic Carbenes as Catalysts in Asymmetric Carbon-Carbon Bond Forming Reactions" |
8:45 pm - 9:30 pm | Jay Siegel (Universität Zürich)
"Topological Stereochemistry" |
THURSDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am -12:30 pm | NEW REACTIONS AND METHODOLOGY |
| Discussion Leader: Lisa Reeder (Pfizer, Inc.) "Stereochemical Features of Some Cyclization Reactions" |
9:00 am - 9:45 am | Tom Hoye (University of Minnesota) |
9:45 am - 10:15 am | Paul Hanson (University of Kansas)
"Multi-Faceted Role of Cyclic Phosphates in Synthesis" |
10:15 am - 10:45 am | Coffee Break |
10:45 am - 11:30 am | William Lubell (University of Montreal)
"Addressing Stereochemical Issues in the Synthesis of Peptide Mimics" |
11:30 am - 12:15 pm | Yadagiri Pendri (Bristol-Myers Squibb)
"Synthesis of Entecavir, a Potent New Antiviral Drug for Hepatitis B" |
12:30 pm | Lunch |
1:30 pm - 6:00 pm | Free Time |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | NOVEL METHODOLOGY |
| Discussion Leader: Erick Carreira (ETH Zürich) |
7:30 pm - 8:15 pm | Patrick Walsh (University of Pennsylvania)
"Asymmetric C-C and C-O Bond Forming Reactions" |
8:15 pm - 9:15 pm | Albert I. Meyers (Colorado State University)
"Chiral Oxazolines: Their Legacy in Asymmetric Synthesis" |
FRIDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am | Departure |