SUNDAY |
4:00 pm - 8:00 pm | Arrival and Check-in (Office Closed 6:00 pm - 7:00 pm) |
6:00 pm | Dinner |
7:30 pm - 7:40 pm | Welcome / Introductory Comments by GRC Site Staff |
7:40 pm - 9:30 pm | Stereoselective Synthesis |
| Discussion Leader: Helma Wennemers (ETH Zurich) |
7:40 pm - 8:25 pm | Yoshito Kishi (Harvard University)
"Natural Product Synthesis" |
8:25 pm - 8:35 pm | Discussion |
8:35 pm - 9:20 pm | Tohru Fukuyama (University of Tokyo)
"Synthetic Studies on Heterocyclic Natural Products" |
9:20 pm - 9:30 pm | Discussion |
MONDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Asymmetric Synthesis |
| Discussion Leader: Anita Mattson (Ohio State University) |
9:00 am - 9:35 am | Jay Siegel (University of Zürich)
"Aromatic Architectures" |
9:35 am - 9:45 am | Discussion |
9:45 am - 10:20 am | Richmond Sarpong (University of California, Berkeley)
"Synthetic Studies Inspired by Complex Alkaloids" |
10:20 am - 10:30 am | Discussion |
10:30 am - 11:00 am | Group Photo / Coffee Break |
11:00 am - 11:35 am | Vy Dong (UC Irvine)
"Stereoselective Strategies for C-H Bond Functionalization" |
11:35 am - 11:45 am | Discussion |
11:45 am - 12:20 pm | Dawei Ma (Shanghai Institute of Organic Chemistry)
"Asymmetric Synthesis of Bioactive Molecules using Organocatalysts" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Stereochemistry in Process R&D |
| Discussion Leader: John Ragan (Pfizer) |
7:30 pm - 8:00 pm | Ian Davies (Merck Research Laboratories)
"What can Steve Jobs Teach us About Stereocontrol?" |
8:00 pm - 8:05 pm | Discussion |
8:05 pm - 8:35 pm | Sèbastien Lemaire (Janssen Pharmaceutica)
"New C-Glycosylation Methodology in the Synthesis of Important Therapeutics" |
8:35 pm - 8:40 pm | Discussion |
8:40 pm - 9:25 pm | Tobias Ritter (Harvard)
|
9:25 pm - 9:30 pm | Discussion |
TUESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Stereoselective Catalysis |
| Discussion Leader: Jon Antilla (Univ. South Florida) |
9:00 am - 9:35 am | Scott Miller (Yale University)
"Stereochemical Aspects of Catalytic Natural Product Modifications" |
9:35 am - 9:45 am | Discussion |
9:45 am - 10:20 am | Pavel Kocovsky (University of Glasgow)
"Organocatalytic Synthesis of Homoallylic Alcohols and their Stereocontrolled Functionalization" |
10:20 am - 10:30 am | Discussion |
10:30 am - 11:00 am | Coffee Break |
11:00 am - 11:35 am | Elizabeth Jarvo (University of California, Irvine)
"Stereospecific Nickel-Catalyzed Cross-Coupling Reactions" |
11:35 am - 11:45 am | Discussion |
11:45 am - 12:20 pm | Matthew Gaunt (University of Cambridge)
"New Copper-Catalyzed Reactions" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Materials and Stereochemistry |
| Discussion Leader: Paul Floreancig (University of Pittsburgh) |
7:30 pm - 8:15 pm | Robert Grubbs (Nobel Laureate, California Institute of Technology)
"Selective metathesis catalysts for the synthesis of molecules and materials" |
8:15 pm - 8:20 pm | Discussion |
8:20 pm - 8:50 pm | David Amabilino (Institut de Ciència de Materials de Barcelona)
"Stereochemistry in nanometer scale aggregates" |
8:50 pm - 8:55 pm | Discussion |
8:55 pm - 9:25 pm | Heather Maynard (UCLA)
"Selective Polymer Conjugations to Enhance Stabilization of Biologic Drugs" |
9:25 pm - 9:30 pm | Discussion |
WEDNESDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Biocatalysis and Enzymology |
| Discussion Leader: Lopa Desai (Bristol-Myers Squibb) |
9:00 am - 9:35 am | Manfred Reetz (Max Planck Institute)
"Laboratory Evolution of Stereoselective Enzymes: A Prolific Source of Catalysts for Asymmetric Reactions" |
9:35 am - 9:45 am | Discussion |
9:45 am - 10:20 am | Nikki Pohl (Iowa State University)
"Carbohydrates" |
10:20 am - 10:30 am | Discussion |
10:30 am - 11:00 am | Coffee Break |
11:00 am - 11:35 am | Daniel Mink (DSM)
"Synthesis of statins by enzymatic C-C bond formation" |
11:35 am - 11:45 am | Discussion |
11:45 am - 12:20 pm | Christina Grozinger (Penn State University)
"Genomics of Chemical Communication in Social Insects" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session |
6:00 pm | Dinner |
7:00 pm - 7:30 pm | Business Meeting |
| Nominations for the next Vice Chair; Fill out Conference Evaluation Forms; Discuss future Site & Scheduling preferences; Election of the next Vice Chair |
7:30 pm - 9:30 pm | Medicinal Stereochemistry |
| Discussion Leader: Scott May (Eli Lilly & Company) |
7:30 pm - 8:15 pm | Steven Ley (University of Cambridge)
"New Tools for Molecule Makers" |
8:15 pm - 8:20 pm | Discussion |
8:20 pm - 8:50 pm | Jacquelyn Gervay-Hague (University of California, Davis)
"Chemically Defined Macromolecular Constructs and Glycolipid Adjuvants in Vaccine Design" |
8:50 pm - 8:55 pm | Discussion |
8:55 pm - 9:25 pm | Punit Seth (Isis Pharmaceuticals)
"Stereochemistry of nucleoside building blocks can modulate the biophysical and biological properties of modified oligonucleotides" |
9:25 pm - 9:30 pm | Discussion |
THURSDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am - 12:30 pm | Stereoselective Synthesis |
| Discussion Leader: Kai Rossen (Sanofi-Aventis) |
9:00 am - 9:35 am | Craig Forsyth (The Ohio State University)
"Stereocontrol in Natural Products Total Synthesis" |
9:35 am - 9:45 am | Discussion |
9:45 am - 10:20 am | Jonathan Reeves (Boehringer Ingelheim)
"New Strategies for Chiral Amine Synthesis" |
10:20 am - 10:30 am | Discussion |
10:30 am - 11:00 am | Coffee Break |
11:00 am - 11:35 am | George Moniz (Eisai Pharmaceuticals)
"Synthesis of Biologically Active Chiral Molecules" |
11:35 am - 11:45 am | Discussion |
11:45 am - 12:20 pm | Jon Rainier (University of Utah)
"Targeting Heterocycles at 4700 Feet above Sea Level" |
12:20 pm - 12:30 pm | Discussion |
12:30 pm | Lunch |
1:30 pm - 4:00 pm | Free Time |
4:00 pm - 6:00 pm | Poster Session |
6:00 pm | Dinner |
7:30 pm - 9:30 pm | Stereoselective Catalysis |
| Discussion Leader: Joel Hawkins (Pfizer) |
7:30 pm - 8:15 pm | Scott Denmark (University of Illinois, Urbana-Champaign)
"Understanding Asymmetric Phase Transfer Catalysis Through Chemoinformatics" |
8:15 pm - 8:25 pm | Discussion |
8:25 pm - 9:10 pm | Ei-ichi Negishi (Nobel Laureate, Purdue University)
"Zr-Catalyzed Asymmetric Carboalumination of Alkenes (ZACA)" |
9:10 pm - 9:20 pm | Discussion |
9:20 pm - 9:30 pm | Closing remarks (Chairs and Future Chairs) |
FRIDAY |
7:30 am - 8:30 am | Breakfast |
9:00 am | Departure |